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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Utah Research Foundation

US Patent
LigandPNGBDBM103924(US8569511, 8)
Affinity DataIC50:  280nMAssay Description:The secondary assay was a time resolved-FRET LanthaScreen Kinase Binding Assay. (Invitrogen Corporation, Carlsbad, Calif.). This assay evaluates the...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Utah Research Foundation

US Patent
LigandPNGBDBM103924(US8569511, 8)
Affinity DataIC50:  300nMAssay Description:Inhibition of PDK1 (unknown origin) after 1 hr in presence of Ser/Thr-07 by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
University Of Utah Research Foundation

US Patent
LigandPNGBDBM103924(US8569511, 8)
Affinity DataIC50:  1.94E+3nMAssay Description:The primary assay for compound inhibitory activity was the ATP depletion assay using the PDKtide substrate purchase from Millipore Corporation.More data for this Ligand-Target Pair
In DepthDetails US Patent