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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetN-acylethanolamine-hydrolyzing acid amidase(Homo sapiens (Human))
Italian Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50151220(CHEMBL3769678)
Affinity DataIC50:  76nMAssay Description:Inhibition of recombinant human NAAA expressed in HEK293 cells after 30 mins by UPLC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-acylethanolamine-hydrolyzing acid amidase(Homo sapiens (Human))
Italian Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50151220(CHEMBL3769678)
Affinity DataIC50:  330nMAssay Description:Inhibition of human BRD3 bromodomain2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid ceramidase(Homo sapiens (Human))
Italian Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50151220(CHEMBL3769678)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of human acid ceramidase by UPLC/MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed