Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50256508(2-(4-((3,3-difluoroazetidin-1-yl)methyl)-2,3-dihyd...)Copy SMILESCopy InChI

Affinity DataEC50:  879nMAssay Description:Agonist activity at human cloned adrenergic alpha1A receptor expressed in CHO cells by calcium mobilization-based fluorescence assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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