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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50155042(2-[2-(5,2'',6''-Trifluoro-biphenyl-3-yl)-2H-tetraz...)
Affinity DataIC50:  108nMAssay Description:In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed