Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019375(4-(4-Benzo[d]isoxazol-3-yl-piperazin-1-yl)-1-(4-fl...)
Affinity DataIC50:  5nMAssay Description:In vitro affinity for cortical alpha-1 adrenergic receptor labelled with [3H]WB-4101More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019375(4-(4-Benzo[d]isoxazol-3-yl-piperazin-1-yl)-1-(4-fl...)
Affinity DataIC50:  69nMAssay Description:In vitro affinity for rat striatal Dopamine receptor D2 labeled with [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed