Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetLong-chain fatty acid transport protein 1(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50433153(CHEMBL2377764)
Affinity DataIC50:  180nMAssay Description:Inhibition of human FLAG-tagged FATP1-mediated [1-14C] oleic acid conversion to [1-14C] oleoyl-CoA after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLong-chain fatty acid transport protein 1(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50433153(CHEMBL2377764)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of mouse FLAG-tagged FATP1-mediated [1-14C] oleic acid conversion to [1-14C] oleoyl-CoA after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed