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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Nuclear receptor ROR-gamma
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50121988
(CHEMBL3617309)
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Affinity Data
EC50: 43nM
Assay Description:
Inverse agonist activity at N-terminal 6xHis-tagged human RORc ligand binding domain (241 to 486) expressed in bacterial expression system assessed a...
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Target Info
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Target
Nuclear receptor ROR-alpha
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50121988
(CHEMBL3617309)
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Affinity Data
EC50: 200nM
Assay Description:
Inverse agonist activity at GAL4-fused human RORa expressed in HEK293 cells assessed as suppression of basal transcriptional activity after 20 hrs by...
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Target Info
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MMDB
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KEGG
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Target
Nuclear receptor ROR-beta
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50121988
(CHEMBL3617309)
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Affinity Data
EC50: 4.10E+3nM
Assay Description:
Inverse agonist activity at GAL4-fused human RORb expressed in HEK293 cells assessed as suppression of basal transcriptional activity after 20 hrs by...
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Target Info
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MMDB
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Target
Nuclear receptor subfamily 1 group I member 2
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50121988
(CHEMBL3617309)
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Affinity Data
EC50: 940nM
Assay Description:
Antagonist activity at GAL4-fused human PXR expressed in HEK293 cells assessed as inhibition of T0901317-stimulated transcriptional activity after 20...
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Target
Oxysterols receptor LXR-alpha
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50121988
(CHEMBL3617309)
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Affinity Data
EC50: 2.60E+3nM
Assay Description:
Antagonist activity at GAL4-fused human LXRalpha expressed in HEK293 cells assessed as inhibition of T0901317-stimulated transcriptional activity aft...
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Target
Oxysterols receptor LXR-beta
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50121988
(CHEMBL3617309)
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Affinity Data
EC50: 3.80E+3nM
Assay Description:
Antagonist activity at GAL4-fused human LXRbeta expressed in HEK293 cells assessed as inhibition of T0901317-stimulated transcriptional activity afte...
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Target
Bile acid receptor
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50121988
(CHEMBL3617309)
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Affinity Data
EC50: 5.90E+3nM
Assay Description:
Antagonist activity at GAL4-fused human FXR expressed in HEK293 cells assessed as inhibition of T0901317-stimulated transcriptional activity after 20...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
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KEGG
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B.MOAD
DrugBank
antibodypedia
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CHEMBL
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In Depth
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Article
PubMed
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Target
Nuclear receptor ROR-gamma
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50121988
(CHEMBL3617309)
Copy SMILES
Copy InChI
Affinity Data
EC50: 3.30E+3nM
Assay Description:
Inverse agonist activity at GAL4-fused human RORc expressed in HEK293 cells assessed as suppression of basal transcriptional activity after 20 hrs by...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
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Article
PubMed
Copy BDB DOI