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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50031053(3-(3,4-Difluoro-phenyl)-indeno[1,2-c]pyridazin-5-o...)
Affinity DataIC50:  5.01nMAssay Description:Inhibition of human supersomes MAOBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50031053(3-(3,4-Difluoro-phenyl)-indeno[1,2-c]pyridazin-5-o...)
Affinity DataIC50:  912nMAssay Description:Inhibition of rat brain MAOBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University Of Geneva

Curated by ChEMBL
LigandPNGBDBM50031053(3-(3,4-Difluoro-phenyl)-indeno[1,2-c]pyridazin-5-o...)
Affinity DataIC50:  920nMAssay Description:Ability to inhibit Monoamine oxidase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50031053(3-(3,4-Difluoro-phenyl)-indeno[1,2-c]pyridazin-5-o...)
Affinity DataIC50:  1.00E+3nMAssay Description:Ability to inhibit Monoamine oxidase A enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed