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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50243107(3-chloro-N-(3-fluorophenyl)benzamide | CHEMBL48624...)
Affinity DataEC50:  297nMAssay Description:Antagonist activity at rat mGluR5 expressed in HEK293A cells assessed as inhibition of glutamate-induced calcium fluorescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed