Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL

LigandBDBM50401908(CHEMBL2207180)Copy SMILESCopy InChI

Affinity DataIC50:  8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Mrc Technology

Curated by ChEMBL

LigandBDBM50401908(CHEMBL2207180)Copy SMILESCopy InChI

Affinity DataIC50:  220nMAssay Description:Inhibition of PDK1 by radiometryMore data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI