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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Cephalon
Curated by
ChEMBL
Ligand
BDBM50361051
(CHEMBL1935590)
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Affinity Data
Ki: 1.60nM
Assay Description:
Displacement of [3H]LSD from full length human 5HT6 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
5-hydroxytryptamine receptor 6
(RAT)
Cephalon
Curated by
ChEMBL
Ligand
BDBM50361051
(CHEMBL1935590)
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Affinity Data
Ki: 6.90nM
Assay Description:
Displacement of [3H]LSD from full length rat 5HT6 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Cephalon
Curated by
ChEMBL
Ligand
BDBM50361051
(CHEMBL1935590)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.60nM
Assay Description:
Antagonist activity at human recombinant 5-HT6 receptor expressed human astrocytoma cells assessed as inhibition of 5-HT-induced cAMP accumulation af...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
Cephalon
Curated by
ChEMBL
Ligand
BDBM50361051
(CHEMBL1935590)
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Affinity Data
IC50: 1.00E+3nM
Assay Description:
Inhibition of human ERG by patch express assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
UniProtKB/TrEMBL
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI