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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Wyeth Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50313143
(5-fluoro-3-(3-fluorophenylsulfonyl)-1-(pyrrolidin-...)
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Affinity Data
Ki: 9.60nM
Assay Description:
Displacement of [3H]LSD from human 5-HT6 receptor expressed in human HeLa cells after 2 hrs
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Wyeth Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50313143
(5-fluoro-3-(3-fluorophenylsulfonyl)-1-(pyrrolidin-...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 38nM
Assay Description:
Agonist activity at human 5-HT6 receptor expressed in human HeLa cells assessed as effect on 5HT-induced intracellular cAMP level after 10 mins by ra...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI