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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50313143(5-fluoro-3-(3-fluorophenylsulfonyl)-1-(pyrrolidin-...)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]LSD from human 5-HT6 receptor expressed in human HeLa cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50313143(5-fluoro-3-(3-fluorophenylsulfonyl)-1-(pyrrolidin-...)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human 5-HT6 receptor expressed in human HeLa cells assessed as effect on 5HT-induced intracellular cAMP level after 10 mins by ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed