Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50071163((2R,4R)-4-Amino-1-(3,4-dichloro-benzyl)-pyrrolidin...)
Affinity DataIC50:  9.90E+4nMAssay Description:In vitro antagonist activity at recombinant Metabotropic glutamate receptor 5 expressed in RGT cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50071163((2R,4R)-4-Amino-1-(3,4-dichloro-benzyl)-pyrrolidin...)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro antagonist activity at recombinant human Metabotropic glutamate receptor 1 expressed in RGT cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed