Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 11 hits in this display
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
Ki: 2.70E+4nMAssay Description:Inhibitory constant of the compound against cloned rat Metabotropic glutamate receptor 1 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
Ki: 4.40E+5nMAssay Description:Inhibitory constant of the compound against cloned rat Metabotropic glutamate receptor 5 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
Ki: >1.00E+6nMAssay Description:Inhibitory constant of the compound against cloned rat Metabotropic glutamate receptor 4 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)
EC50: >1.00E+6nMAssay Description:Activity of the compound tested at cloned rat Metabotropic glutamate receptor 4 expressed in Chinese Hamster Ovary (CHO) cellsMore data for this Ligand-Target Pair
BDBM50130515((3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclo...)