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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50407826
(CHEMBL2114105)
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Affinity Data
Ki: >2.70E+5nM
Assay Description:
Binding affinity towards metabotropic glutamate receptor mGluR1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50407826
(CHEMBL2114105)
Copy SMILES
Copy InChI
Affinity Data
Ki: >2.80E+5nM
Assay Description:
Binding affinity of the compound towards metabotropic glutamate receptor mGluR4a
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50407826
(CHEMBL2114105)
Copy SMILES
Copy InChI
Affinity Data
IC50: >3.00E+5nM
Assay Description:
Concentration required for the half-maximal inhibition of PI hydrolysis in BHK cells expressing mGluR1a
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50407826
(CHEMBL2114105)
Copy SMILES
Copy InChI
Affinity Data
IC50: >3.00E+5nM
Assay Description:
Concentration required for the half-maximal inhibition of cAMP hydrolysis in BHK cells expressing mGluR2
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50407826
(CHEMBL2114105)
Copy SMILES
Copy InChI
Affinity Data
IC50: >3.00E+5nM
Assay Description:
Concentration required for the half-maximal inhibition of cAMP hydrolysis in BHK cells expressing mGluR4
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50407826
(CHEMBL2114105)
Copy SMILES
Copy InChI
Affinity Data
EC50: >3.00E+5nM
Assay Description:
Effective concentration forskolin-stimulated cAMP formation in BHK cells expressing mGluR2 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50407826
(CHEMBL2114105)
Copy SMILES
Copy InChI
Affinity Data
EC50: >3.00E+5nM
Assay Description:
Concentration required for half-maximal stimulation of PI hydrolysis in BHK cells expressing mGluR1a
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50407826
(CHEMBL2114105)
Copy SMILES
Copy InChI
Affinity Data
EC50: >3.00E+5nM
Assay Description:
Effective concentration against forskolin-stimulated cAMP formation in BHK cells expressing mGluR4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI