Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50407828(CHEMBL2114106)
Affinity DataKi: >2.70E+5nMAssay Description:Binding affinity towards metabotropic glutamate receptor mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50407828(CHEMBL2114106)
Affinity DataKi: >2.80E+5nMAssay Description:Binding affinity of the compound towards metabotropic glutamate receptor mGluR4aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50407828(CHEMBL2114106)
Affinity DataIC50: >3.00E+5nMAssay Description:Concentration required for the half-maximal inhibition of PI hydrolysis in BHK cells expressing mGluR1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50407828(CHEMBL2114106)
Affinity DataIC50: >3.00E+5nMAssay Description:Concentration required for the half-maximal inhibition of cAMP hydrolysis in BHK cells expressing mGluR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50407828(CHEMBL2114106)
Affinity DataIC50: >3.00E+5nMAssay Description:Concentration required for the half-maximal inhibition of cAMP hydrolysis in BHK cells expressing mGluR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50407828(CHEMBL2114106)
Affinity DataEC50: >3.00E+5nMAssay Description:Effective concentration forskolin-stimulated cAMP formation in BHK cells expressing mGluR2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50407828(CHEMBL2114106)
Affinity DataEC50: >3.00E+5nMAssay Description:Concentration required for half-maximal stimulation of PI hydrolysis in BHK cells expressing mGluR1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50407828(CHEMBL2114106)
Affinity DataEC50: >3.00E+5nMAssay Description:Effective concentration against forskolin-stimulated cAMP formation in BHK cells expressing mGluR4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed