Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

Curated by ChEMBL

LigandBDBM50351025(CHEMBL1819324)Copy SMILESCopy InChI

Affinity DataIC50:  4.22E+4nMAssay Description:Inhibition of pig kidney microsomal APN assessed as hydrolysis of L-Leu-p-nitroanilide after 1 hr by spectrophotometryMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

Curated by ChEMBL

LigandBDBM50351025(CHEMBL1819324)Copy SMILESCopy InChI

Affinity DataIC50:  6.74E+4nMAssay Description:Inhibition of human MMP-2 after 30 mins by spectrophotometryMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI