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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
University Of Cagliari
Curated by
ChEMBL
Ligand
BDBM50324021
((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
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Affinity Data
Ki: 1.01nM
Assay Description:
Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
University Of Cagliari
Curated by
ChEMBL
Ligand
BDBM50324021
((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
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Affinity Data
Ki: 54.5nM
Assay Description:
Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(MOUSE)
University Of Cagliari
Curated by
ChEMBL
Ligand
BDBM50324021
((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
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Affinity Data
IC50: 67.3nM
Assay Description:
Agonist activity at delta opioid receptor in mouse vas deference
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Cagliari
Curated by
ChEMBL
Ligand
BDBM50324021
((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
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Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Agonist activity at mu opioid receptor in Hartley guinea pig small intestine
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI