Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205831(CHEMBL387159 | H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylg...)
Affinity DataKi:  2.34nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205831(CHEMBL387159 | H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylg...)
Affinity DataKi:  5.87nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205831(CHEMBL387159 | H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylg...)
Affinity DataKi:  309nMAssay Description:Displacement of [3H]U69,593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205831(CHEMBL387159 | H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylg...)
Affinity DataIC50:  1.02nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205831(CHEMBL387159 | H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylg...)
Affinity DataIC50:  3.19nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed