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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by
ChEMBL
Ligand
BDBM50018635
(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
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Affinity Data
Ki: 22nM
Assay Description:
Binding affinity towards Opioid receptor mu 1 in rat brain membrane using [3H]-DAGO as radioligand
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by
ChEMBL
Ligand
BDBM50018635
(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
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Copy InChI
Affinity Data
Ki: 422nM
Assay Description:
Inhibition of [3H]-DSLET binding to rat brain membrane Opioid receptor delta 1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(GUINEA PIG)
Clinical Research Institute Of Montreal
Curated by
ChEMBL
Ligand
BDBM50018635
(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
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Affinity Data
IC50: 632nM
Assay Description:
Inhibitory activity towards electrically induced contractions in guinea pig ileum expressing Opioid receptor mu 1
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(MOUSE)
Clinical Research Institute Of Montreal
Curated by
ChEMBL
Ligand
BDBM50018635
(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2...)
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Copy InChI
Affinity Data
IC50: 4.81E+3nM
Assay Description:
Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI