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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by
ChEMBL
Ligand
BDBM50205832
(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
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Affinity Data
Ki: 0.550nM
Assay Description:
Displacement of [3H]DAMGO from rat brain mu opioid receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by
ChEMBL
Ligand
BDBM50205832
(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
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Copy InChI
Affinity Data
Ki: 0.822nM
Assay Description:
Displacement of [3H]DSLET from rat brain delta opioid receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal
Curated by
ChEMBL
Ligand
BDBM50205832
(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
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Affinity Data
Ki: 44.9nM
Assay Description:
Displacement of [3H]U69,593 from guinea pig brain kappa opioid receptor
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(MOUSE)
Clinical Research Institute Of Montreal
Curated by
ChEMBL
Ligand
BDBM50205832
(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
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Affinity Data
IC50: 0.562nM
Assay Description:
Agonist activity at delta opioid receptor in mouse vas deferens
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(GUINEA PIG)
Clinical Research Institute Of Montreal
Curated by
ChEMBL
Ligand
BDBM50205832
(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
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Copy InChI
Affinity Data
IC50: 1.30nM
Assay Description:
Agonist activity at mu opioid receptor in guinea pig ileum
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI