Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
Affinity DataKi:  0.822nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
Affinity DataKi:  44.9nMAssay Description:Displacement of [3H]U69,593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
Affinity DataIC50:  0.562nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(CHEMBL220327 | H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2)
Affinity DataIC50:  1.30nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed