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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50295263
((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
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Affinity Data
Ki: 2.30nM
Assay Description:
Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50295263
((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
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Copy InChI
Affinity Data
Ki: 3.50E+3nM
Assay Description:
Displacement of [3H]DPDE from delta opioid receptor in rat brain membrane by liquid scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(GUINEA PIG)
Universit£
Curated by
ChEMBL
Ligand
BDBM50295263
((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
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Affinity Data
IC50: 7.90E+3nM
Assay Description:
Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated contraction
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(MOUSE)
Universit£
Curated by
ChEMBL
Ligand
BDBM50295263
((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
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Copy InChI
Affinity Data
IC50: 1.40E+5nM
Assay Description:
Agonist activity at delta opioid receptor in mouse vas deference assessed as inhibition of electrically-stimulated contraction
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI