Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMu-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326890((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataKi:  510nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326890((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataKi:  6.30E+3nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50326890((S)-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((...)
Affinity DataIC50:  2.70E+3nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed