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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50166124((S)-2-{(R)-2-[(S)-2-Amino-3-(3H-imidazol-4-yl)-pro...)
Affinity DataEC50:  67nMAssay Description:In vitro agonist potency for Mouse Melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50166124((S)-2-{(R)-2-[(S)-2-Amino-3-(3H-imidazol-4-yl)-pro...)
Affinity DataEC50:  250nMAssay Description:In vitro agonist potency for Mouse Melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50166124((S)-2-{(R)-2-[(S)-2-Amino-3-(3H-imidazol-4-yl)-pro...)
Affinity DataEC50:  2.78nMAssay Description:In vitro agonist potency for Mouse Melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50166124((S)-2-{(R)-2-[(S)-2-Amino-3-(3H-imidazol-4-yl)-pro...)
Affinity DataEC50:  18.5nMAssay Description:In vitro agonist potency for Mouse Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed