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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Glutamate receptor ionotropic, kainate 2
(Rattus norvegicus)
University Walk
Curated by
ChEMBL
Ligand
BDBM50178145
((S)-1-(2-amino-2-carboxyethyl)-3-(2-carboxybenzyl)...)
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Affinity Data
Ki: >1.00E+5nM
Assay Description:
Displacement of [3H]kainate from rat GLUK6 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Glutamate receptor ionotropic, kainate 1
(RAT)
University Walk
Curated by
ChEMBL
Ligand
BDBM50178145
((S)-1-(2-amino-2-carboxyethyl)-3-(2-carboxybenzyl)...)
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Copy InChI
Affinity Data
Kd: 209nM
Assay Description:
Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibres
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor ionotropic, kainate 1
(RAT)
University Walk
Curated by
ChEMBL
Ligand
BDBM50178145
((S)-1-(2-amino-2-carboxyethyl)-3-(2-carboxybenzyl)...)
Copy SMILES
Copy InChI
Affinity Data
Kd: 209nM
Assay Description:
Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibers
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI