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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Glutamate receptor ionotropic, kainate 2
(Rattus norvegicus)
University Walk
Curated by
ChEMBL
Ligand
BDBM50178138
((S)-1-(2-amino-2-carboxyethyl)-3-(2-carboxyethyl)p...)
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Affinity Data
Ki: >1.00E+5nM
Assay Description:
Displacement of [3H]kainate from rat GLUK6 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
MMDB
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor ionotropic, kainate 2
(Rattus norvegicus)
University Walk
Curated by
ChEMBL
Ligand
BDBM50178138
((S)-1-(2-amino-2-carboxyethyl)-3-(2-carboxyethyl)p...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+6nM
Assay Description:
Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
MMDB
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor ionotropic, kainate 1
(RAT)
University Walk
Curated by
ChEMBL
Ligand
BDBM50178138
((S)-1-(2-amino-2-carboxyethyl)-3-(2-carboxyethyl)p...)
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Copy InChI
Affinity Data
Kd: 7.31E+4nM
Assay Description:
Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibers
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
MMDB
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor ionotropic, kainate 5
(Rattus norvegicus)
University Walk
Curated by
ChEMBL
Ligand
BDBM50178138
((S)-1-(2-amino-2-carboxyethyl)-3-(2-carboxyethyl)p...)
Copy SMILES
Copy InChI
Affinity Data
Kd: 7.31E+4nM
Assay Description:
Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibers
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
MMDB
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI