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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
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kcal/mol
)
Found
2
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Target
Aminopeptidase N
(Sus scrofa (Pig))
Shandong University
Ligand
BDBM240828
((2R,3S)-3-amino-2-hydroxy-N-((S)-2-(hydroxyamino)-...)
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Affinity Data
IC50: 1.26E+3nM
pH: 7.5 T: 2°C
Assay Description:
IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
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Article
PubMed
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Target
72 kDa type IV collagenase
(Sus scrofa (Pig))
Shandong University
Ligand
BDBM240828
((2R,3S)-3-amino-2-hydroxy-N-((S)-2-(hydroxyamino)-...)
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Affinity Data
IC50: 2.13E+5nM
Assay Description:
Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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