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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

LigandPNGBDBM240828((2R,3S)-3-amino-2-hydroxy-N-((S)-2-(hydroxyamino)-...)
Affinity DataIC50:  1.26E+3nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Sus scrofa (Pig))
Shandong University

LigandPNGBDBM240828((2R,3S)-3-amino-2-hydroxy-N-((S)-2-(hydroxyamino)-...)
Affinity DataIC50:  2.13E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed