Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068512((1S,2R)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  21.3nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068512((1S,2R)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  93.5nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068512((1S,2R)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  132nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068512((1S,2R)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  810nMAssay Description:Binding affinity against the 5-hydroxytryptamine 1A receptor labelled with [3H]-8-OH-DPAT in rat hippocampal homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed