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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetCorticotropin-releasing factor receptor 2(Mus musculus)
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403726(CHEMBL2112936)
Affinity DataKi:  20nMAssay Description:Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 2 betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403726(CHEMBL2112936)
Affinity DataKi:  110nMAssay Description:Antagonistic activity against [125I]-Tyr-ovine CRF binding to Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403726(CHEMBL2112936)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403726(CHEMBL2112936)
Affinity DataKi:  3.20E+3nMAssay Description:Binding affinity against dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403726(CHEMBL2112936)
Affinity DataKi:  4.20E+3nMAssay Description:Binding affinity against Neuropeptide Y receptor type 1 using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Agouron Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403726(CHEMBL2112936)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed