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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Tyrosine-protein kinase SYK
(Homo sapiens (Human))
Taiho Pharmaceutical
US Patent
Ligand
BDBM182797
(US9145414, 160)
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Affinity Data
IC50: 0.380nM
pH: 7.5 T: 2°C
Assay Description:
The in vitro inhibitory activity of the compound of the present invention against Syk kinase activity was assayed under the following conditions: the...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
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Target
Aurora kinase B
(Homo sapiens (Human))
Taiho Pharmaceutical
US Patent
Ligand
BDBM182797
(US9145414, 160)
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Affinity Data
IC50: 1.30E+3nM
pH: 7.4 T: 2°C
Assay Description:
The in vitro inhibitory activity of the compound against Aurora B kinase activity was assayed with reference to a method described in patent publicat...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Taiho Pharmaceutical
US Patent
Ligand
BDBM182797
(US9145414, 160)
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Affinity Data
IC50: 1.40E+3nM
pH: 7.5
Assay Description:
Conditions for assaying the in vitro inhibitory activity of the compound against KDR kinase activity were set with reference to the statement in the ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI