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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by
ChEMBL
Ligand
BDBM50186367
(CHEMBL379959 | c(his-D-phe-arg-trp-Ahp))
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Affinity Data
Ki: 244nM
Assay Description:
Displacement of [125I]NDP-alpha-MSH from human cloned MC4R expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by
ChEMBL
Ligand
BDBM50186367
(CHEMBL379959 | c(his-D-phe-arg-trp-Ahp))
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Copy InChI
Affinity Data
EC50: 67nM
Assay Description:
Activity at human MC1R by cAMP accumulation in SaoS2 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Asahi Kasei Pharma
Curated by
ChEMBL
Ligand
BDBM50186367
(CHEMBL379959 | c(his-D-phe-arg-trp-Ahp))
Copy SMILES
Copy InChI
Affinity Data
EC50: 15.4nM
Assay Description:
Activity at human MC4R by cAMP accumulation in SaoS2 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI