Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50127296((R)-3-[(S)-5-(3-Guanidino-propylcarbamoyl)-2-oxo-1...)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of fibronectin (GST-3Fn8-11) binding to recombinant soluble mini integrin alpha5-beta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50127297(3-[5-(3-Guanidino-propylcarbamoyl)-2-oxo-1-aza-bic...)
Affinity DataIC50:  1.30E+6nMAssay Description:Inhibition of fibronectin (GST-3Fn8-11) binding to recombinant soluble mini integrin alpha5-beta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50127298((R)-3-[(R)-5-(3-Guanidino-propylcarbamoyl)-2-oxo-1...)
Affinity DataIC50:  3.10E+6nMAssay Description:Inhibition of fibronectin (GST-3Fn8-11) binding to recombinant soluble mini integrin alpha5-beta1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed