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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Mu-type opioid receptor
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50219924
(6-[4-(phenethylamino-methyl)-phenoxy]-nicotinamidi...)
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Affinity Data
Ki: 21nM
Assay Description:
Antagonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assay
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50219924
(6-[4-(phenethylamino-methyl)-phenoxy]-nicotinamidi...)
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Copy InChI
Affinity Data
Ki: 215nM
Assay Description:
Displacement of [3H]bremazocine from human delta opioid receptor expressed in CHO cells in presence of high sodium by SPA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50219924
(6-[4-(phenethylamino-methyl)-phenoxy]-nicotinamidi...)
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Copy InChI
Affinity Data
Ki: 1.15E+3nM
Assay Description:
Displacement of [3H]diprenorphine from human kappa opioid receptor expressed in CHO cells in presence of high sodium by SPA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI