Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101527((R)-3-(((S)-1-amino-3-cyclohexyl-1-oxopropan-2-yl)...)
Affinity DataKi:  123nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101527((R)-3-(((S)-1-amino-3-cyclohexyl-1-oxopropan-2-yl)...)
Affinity DataKi:  123nMAssay Description:Inhibitory constant against matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101527((R)-3-(((S)-1-amino-3-cyclohexyl-1-oxopropan-2-yl)...)
Affinity DataKi:  3.12E+3nMAssay Description:Inhibition of the Stromelysin enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101527((R)-3-(((S)-1-amino-3-cyclohexyl-1-oxopropan-2-yl)...)
Affinity DataKi:  3.12E+3nMAssay Description:Inhibitory constant against matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50101527((R)-3-(((S)-1-amino-3-cyclohexyl-1-oxopropan-2-yl)...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50101527((R)-3-(((S)-1-amino-3-cyclohexyl-1-oxopropan-2-yl)...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibitory constant against matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50101527((R)-3-(((S)-1-amino-3-cyclohexyl-1-oxopropan-2-yl)...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of the Collagenase enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article