Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50111197((S)-2-[(1H-Indol-3-ylmethyl)-amino]-3-naphthalen-2...)
Affinity DataKi:  2.60E+4nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50111197((S)-2-[(1H-Indol-3-ylmethyl)-amino]-3-naphthalen-2...)
Affinity DataKi:  6.00E+4nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50111197((S)-2-[(1H-Indol-3-ylmethyl)-amino]-3-naphthalen-2...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50111197((S)-2-[(1H-Indol-3-ylmethyl)-amino]-3-naphthalen-2...)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity in competition with [125I]NDP-MSH on recombinant melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed