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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Substance-P receptor
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50283777
(BDBM50284761 | CHEMBL295022 | CHEMBL32248 | [1-(1-...)
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Affinity Data
IC50: 4.20E+3nM
Assay Description:
Inhibitory activity against binding of [125I]-Bolton-Hunter SP to tachykinin NK-1 receptor in human lymphoma IM9 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
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Target
Substance-K receptor
(HAMSTER)
TBA
Curated by
ChEMBL
Ligand
BDBM50283777
(BDBM50284761 | CHEMBL295022 | CHEMBL32248 | [1-(1-...)
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Affinity Data
IC50: 5.20E+3nM
Assay Description:
Binding affinity towards Tachykinin receptor 2 using [125I]iodohistidyl-NKA (0.1 nM)) as radioligand
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
Target
Substance-P receptor
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50283777
(BDBM50284761 | CHEMBL295022 | CHEMBL32248 | [1-(1-...)
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Copy InChI
Affinity Data
IC50: 9.30E+3nM
Assay Description:
Inhibition of [125I]-BH-SP binding to tachykinin NK1 receptor in human IM-9 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI
Target
Neuromedin-K receptor
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50283777
(BDBM50284761 | CHEMBL295022 | CHEMBL32248 | [1-(1-...)
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Copy InChI
Affinity Data
IC50: 9.30E+3nM
Assay Description:
Binding affinity towards Tachykinin receptor 3 using [125I]-[Mephe7] NKB as radioligand
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI