Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283777(BDBM50284761 | CHEMBL295022 | CHEMBL32248 | [1-(1-...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibitory activity against binding of [125I]-Bolton-Hunter SP to tachykinin NK-1 receptor in human lymphoma IM9 cellsMore data for this Ligand-Target Pair
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TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50283777(BDBM50284761 | CHEMBL295022 | CHEMBL32248 | [1-(1-...)
Affinity DataIC50:  5.20E+3nMAssay Description:Binding affinity towards Tachykinin receptor 2 using [125I]iodohistidyl-NKA (0.1 nM)) as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283777(BDBM50284761 | CHEMBL295022 | CHEMBL32248 | [1-(1-...)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of [125I]-BH-SP binding to tachykinin NK1 receptor in human IM-9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283777(BDBM50284761 | CHEMBL295022 | CHEMBL32248 | [1-(1-...)
Affinity DataIC50:  9.30E+3nMAssay Description:Binding affinity towards Tachykinin receptor 3 using [125I]-[Mephe7] NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article