Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
3-phosphoinositide-dependent protein kinase 1
(Homo sapiens (Human))
Merck Patent
US Patent
Ligand
BDBM116994
(US8637532, 721)
Copy SMILES
Copy InChI
Affinity Data
IC50: 60nM
pH: 7.5 T: 2°C
Assay Description:
The kinase assay is performed as 384-well Flashplate assay (PerkinElmer LAS Germany GmbH). 3.4 nM His6-PDK1(Delta 1-50) (PDK1 that has a His-tag cons...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Ribosomal protein S6 kinase beta-1
(Homo sapiens (Human))
Merck Patent
US Patent
Ligand
BDBM116994
(US8637532, 721)
Copy SMILES
Copy InChI
Affinity Data
IC50: 700nM
pH: 7.5 T: 2°C
Assay Description:
P70S6K inhibitor compounds are diluted and plated in 96 well plates. A reaction mixture including the following components is then added to the compo...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI