Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMelanocortin receptor 4(Homo sapiens (Human))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374670(CHEMBL270923)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]NDP-alpha-MSH from MC4RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374670(CHEMBL270923)
Affinity DataEC50:  550nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374670(CHEMBL270923)
Affinity DataEC50:  390nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374670(CHEMBL270923)
Affinity DataEC50:  150nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
The Hebrew University Of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50374670(CHEMBL270923)
Affinity DataEC50:  2.05E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed