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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
119
hits in this display
Target
Fatty-acid amide hydrolase 1
(Mus musculus (mouse))
Universit£
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
Ki: 1.20nM
Assay Description:
Inhibition of mouse FAAH isolated from brain homogenate using [3H-ethanolamine]AEA as substrate incubated for 20 mins prior to substrate addition mea...
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Target
Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
Ki: 2.00E+3nM
Assay Description:
Enzyme-coupled assay using oleamide as substrate where stoichiometic quantites of NAD are formed upon the generation of ammonia from oleamide by FAAH...
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Target
5-hydroxytryptamine receptor 1E
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
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Target
Alpha-2A adrenergic receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
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Target
Alpha-2B adrenergic receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
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Target
Alpha-2C adrenergic receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
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Target
Beta-1 adrenergic receptor
(Rattus norvegicus (Rat))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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Target
Beta-2 adrenergic receptor
(Rattus norvegicus)
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
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Target
Cannabinoid receptor 1
(Rattus norvegicus (rat))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
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Target
Cannabinoid receptor 2
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
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Target
Muscarinic acetylcholine receptor M2
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
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CHEMBL
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Target
Muscarinic acetylcholine receptor M3
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
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CHEMBL
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Target
Muscarinic acetylcholine receptor M4
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
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Target
Muscarinic acetylcholine receptor M5
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
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Target
Neuronal acetylcholine receptor subunit alpha-2
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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Target
Neuronal acetylcholine receptor subunit alpha-2
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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Target
Neuronal acetylcholine receptor subunit alpha-3
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
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CHEMBL
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Target
Neuronal acetylcholine receptor subunit alpha-3
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
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Target
Neuronal acetylcholine receptor subunit alpha-4
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
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GoogleScholar
Ligand Info
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CHEMBL
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Article
PubMed
Copy BDB DOI
Target
Neuronal acetylcholine receptor subunit alpha-4
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
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GoogleScholar
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CHEMBL
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Article
PubMed
Copy BDB DOI
Target
D(1A) dopamine receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
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Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
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Target
D(1B) dopamine receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
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Target
Sodium-dependent dopamine transporter
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
NCI pathway
Reactome pathway
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Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
UniProtKB/TrEMBL
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Target
Histamine H1 receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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Target
Histamine H2 receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
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GoogleScholar
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CHEMBL
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ATP-dependent translocase ABCB1
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Ki: >1.00E+4nM
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Sodium-dependent noradrenaline transporter
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Ki: >1.00E+4nM
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Kappa-type opioid receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Ki: >1.00E+4nM
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Mu-type opioid receptor
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Ki: >1.00E+4nM
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Sigma non-opioid intracellular receptor 1
(RAT)
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Ki: >1.00E+4nM
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AP-2 complex subunit sigma
(RAT)
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Ki: >1.00E+4nM
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5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Ki: >1.00E+4nM
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5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
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Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
Ki: >1.00E+4nM
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Mcgill University
Curated by
PDSP K
i
Database
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Ki: >1.00E+4nM
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 0.240nM
Assay Description:
Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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IC50: 0.5nM
Assay Description:
Inhibition of rat intact neuron FAAH
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 0.5nM
Assay Description:
Inhibition of FAAH in Wistar rat brain intact neurons assessed as reduction in [3H]anandamide hydrolysis using [3H]anandamide as substrate preincubat...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 1.20nM
pH: 7.6 T: 2°C
Assay Description:
In this assay, 0.05 Units of hFAAH was pre-incubated for 30 min at 37 C with 2 uL of 11a, 11b, 11f at different concentrations (0.01 - 100 uM) or veh...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 1.70nM
Assay Description:
Inhibition of FAAH in Sprague-Dawley rat brain homogenates preincubated for 10 mins followed by addition of substrate measured after 30 mins by liqui...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 3nM
Assay Description:
Inhibition of rat FAAH assessed as hydrolysis of anandamidoaminomethylcumarin
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 3.80nM
Assay Description:
Inhibition of Wistar rat brain FAAH
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 3.80nM
Assay Description:
Inhibition of FAAH (unknown origin)
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 3.80nM
Assay Description:
Inhibition of FAAH in Wistar rat cerebral membrane by liquid scintillation counting
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 4nM
Assay Description:
Inhibition of human FAAH assessed as hydrolysis of anandamidoaminomethylcumarin
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 4nM
Assay Description:
Inhibition of FAAH (unknown origin)
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 4.57nM
Assay Description:
Displacement of [3H]-anandamide from rat brain FAAH after 30 mins by scintillation counting
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of FAAH in rat brain membrane using anandamide[ethanolamine-3H] as substrate assessed as reduction in [3H]-ethanolamine production incubat...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of FAAH in rat brain membrane assessed as [3H]anandamide hydrolysis
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of FAAH
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of FAAH in Wistar rat brain membranes assessed as reduction in [3H]anandamide hydrolysis using [3H]anandamide as substrate preincubated fo...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting method
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Target
Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of FAAH in Wistar rat brain membranes using [3H]-anandamide as substrate preincubated for 10 mins followed by substrate addition measured ...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Displacement of [3H]anandamide from FAAH in rat brain membranes after 30 mins by liquid scintillation counting
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of human FAAH
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Target
Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of [3H]-anandamide binding to fatty acid amide hydrolase of rat brain membranes
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Fatty-acid amide hydrolase 1
(Mus musculus (mouse))
Universit£
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of mouse FAAH isolated from brain homogenate using [3H-ethanolamine]AEA as substrate incubated for 20 mins prior to substrate addition mea...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 4.60nM
Assay Description:
Irreversible inhibition of human recombinant FAAH assessed as hydrolysis of [3H]-AEA after 10 mins by liquid scintillation counting
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of rat brain membrane FAAH
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.60nM
Assay Description:
Inhibition of FAAH
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Target
Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 4.90nM
Assay Description:
Inhibition of rat histidine tagged FAAH expressed in Escherichia coli by coumarin ester substrate fluorescence assay
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Fatty-acid amide hydrolase 2
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 5nM
Assay Description:
Inhibition of recombinant human N-terminal FLAG-tagged/C-terminal Myc-His6 tagged FAAH2 (32 to 579 residues) expressed in COS7 cell membranes
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 6nM
Assay Description:
Inhibition of FAAH in rat brain membranes assessed as hydrolysis of [14C]-anandamide preincubated for 20 mins before [14C]-anandamide addition measur...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 6.90nM
Assay Description:
Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate preincubated with protein for 60 mins followed by substrate addition b...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 7.70nM
Assay Description:
The assays for compounds described herein are amenable to high throughput screening. Preferred assays thus detect binding of the inhibitor to FAAH or...
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Fatty-acid amide hydrolase 1
(Mus musculus (mouse))
Universit£
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 11nM
Assay Description:
Inhibition of FAAH in mouse brain microsomes using OMP substrate by fluorescence based assay
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 12nM
Assay Description:
Inhibition of FAAH in rat brain microsomes using OMP substrate by fluorescence based assay
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 13nM
Assay Description:
Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate preincubated with protein for 30 mins followed by substrate addition b...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 15nM
Assay Description:
Inhibition of human recombinant FAAH expressed in Escherichia coli assessed as hydrolysis of [3H]-AEA
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 18nM
Assay Description:
Inhibition of rat brain FAAH using [3H]AEA as substrate preincubated for 10 mins at pH 8
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 22nM
Assay Description:
Inhibition of rat FAAH incubated 3 hrs prior to addition of arachidonylaminomethylcoumarin amide
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 23nM
Assay Description:
Inhibition of human FAAH expressed in baculovirus-infected High Five cells S9 fraction using OMP substrate by fluorescence based assay
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 24nM
pH: 9.0
Assay Description:
Inhibition of FAAH in rat brain membrane at pH 9 using N-arachidonoyl-[14C]-ethanolamine as substrate preincubated for 10 mins followed by substrate ...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 32nM
Assay Description:
Inhibition of human FAAH using N-(6-methoxypyridin-3-yl)octanamide as a substrate assessed as reduction in 6-methoxypyridin-3-amine formation by fluo...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 40nM
Assay Description:
Inhibition of human recombinant FAAH expressed in Escherichia coli using [3H]AEA substrate incubated at 37 degC for 10 mins by liquid scintillation c...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 43nM
Assay Description:
Inhibition of FAAH in rat brain membrane using N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide as substrate measured after 60 mins by reverse-phase HPLC-ba...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 48nM
Assay Description:
Inhibition of rat FAAH preincubated for 20 mins
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 58nM
Assay Description:
Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate preincubated with protein for 0 min followed by substrate addition by ...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Copy InChI
Affinity Data
IC50: 59nM
Assay Description:
Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate after 30 mins by fluorescence assay
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Copy InChI
Affinity Data
IC50: 60nM
Assay Description:
Inhibition of FAAH in rat brain microsomes using N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide as substrate after 60 mins by fluorescence-based HPLC anal...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 60nM
Assay Description:
Inhibition of FAAH in rat brain microsomes using N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide as substrate after 60 mins by fluorescence-based reversed ...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 62nM
Assay Description:
Inhibition of FAAH in Sprague-Dawley rat brain microsomes assessed as N-(2-hydroxyethyl)-4-pyren-1-ylbutanamide conversion to 4-pyren-1-ylbutanoic ac...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 63nM
Assay Description:
Inhibition of rat FAAH incubated 1 hr prior to addition of arachidonylaminomethylcoumarin amide
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
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Affinity Data
IC50: 64nM
Assay Description:
Inhibition of rat brain FAAH using [3H]AEA as substrate preincubated for 10 mins at pH 6
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 67nM
Assay Description:
Inhibition of Sprague-Dawley rat brain microsome FAAH assessed as reduction in 4-pyren-1-ylbutanoic acid release after 60 mins by reverse phase HPLC-...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 78nM
Assay Description:
Inhibition of human FAAH incubated 1 hr prior to addition of arachidonylaminomethylcoumarin amide
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 90nM
Assay Description:
Inhibition of human recombinant FAAH in assessed as hydrolysis of [14C]-anandamide preincubated for 20 mins before [14C]-anandamide addition measured...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 109nM
Assay Description:
Inhibition of recombinant human N-terminal -His6 tagged FAAH (32 to 579 residues) expressed in Escherichia coli BL21 preincubated for 60 mins followe...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 109nM
pH: 7.4 T: 2°C
Assay Description:
FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 109nM
Assay Description:
Inhibition of FAAH
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Fatty-acid amide hydrolase 1
(Mus musculus (mouse))
Universit£
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ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 110nM
Assay Description:
Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting method
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 141nM
pH: 7.4
Assay Description:
Inhibition of FAAH in rat brain membrane at pH 7.4 using N-arachidonoyl-[14C]-ethanolamine as substrate preincubated for 10 mins followed by substrat...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 166nM
Assay Description:
Inhibition of human recombinant FAAH overexpressed in African green monkey COS7 cells using [3H]-anandamide as substrate preincubated for 10 mins bef...
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 170nM
Assay Description:
Inhibition of human recombinant FAAH overexpressed in African green monkey COS7 cells using [3H]-anandamide as substrate preincubated for 10 mins bef...
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Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
Pfizer
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 240nM
Assay Description:
Inhibition of FAAH from rat brain microsomes by RP-HPLC
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Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 260nM
Assay Description:
Inhibition of human recombinant FAAH expressed in sf21 cells using AMC-AA as substrate preincubated for 15 mins followed by substrate addition measur...
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Target
Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 572nM
pH: 7.4 T: 2°C
Assay Description:
FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o...
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Copy BDB DOI
Target
Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Copy InChI
Affinity Data
IC50: 856nM
pH: 7.4 T: 2°C
Assay Description:
FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o...
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Copy BDB DOI
Target
Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Copy InChI
Affinity Data
IC50: 986nM
Assay Description:
Inhibition of recombinant human N-terminal -His6 tagged FAAH (32 to 579 residues) expressed in Escherichia coli BL21-AI preincubated for 5 mins follo...
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Copy BDB DOI
Target
Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
E.I. Du Pont De Nemours
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 986nM
pH: 7.4 T: 2°C
Assay Description:
FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o...
More data for this Ligand-Target Pair
Target Info
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Target
Bifunctional epoxide hydrolase 2
(Homo sapiens (Human))
University Of California Davis
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: 1.10E+3nM
Assay Description:
Inhibition of human recombinant soluble epoxide hydrolase expressed in baculovirus-infected High Five cells S9 fraction using CMNPC substrate by fluo...
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Target
Prostaglandin G/H synthase 2
(Homo sapiens (Human))
Fondazione Istituto Italiano Di Tecnologia
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of recombinant human COX2 assessed as production of PGF2-alpha preincubated with compound followed by the addition of 5 uM arachidonic aci...
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Prostaglandin G/H synthase 1
(Ovis aries (Sheep))
Fondazione Istituto Italiano Di Tecnologia
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of ovine COX1 assessed as production of PGF2-alpha preincubated with compound followed by the addition of 5 uM arachidonic acid as substra...
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Transient receptor potential cation channel subfamily A member 1
(Homo sapiens (Human))
Ferrara University
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
EC50: 2.45E+4nM
Assay Description:
Agonist activity at human TRPA1 channel expressed in HEK293 cells assessed as increase in intracellular calcium influx
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Transient receptor potential cation channel subfamily A member 1
(Homo sapiens (Human))
Ferrara University
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
EC50: 1.34E+8nM
Assay Description:
Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assay
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Copy BDB DOI
Target
Transient receptor potential cation channel subfamily A member 1
(Homo sapiens (Human))
Ferrara University
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
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Affinity Data
EC50: 2.45E+4nM
Assay Description:
Agonist activity at human TRPA1 expressed in HEK293F cells assessed as increase in calcium influx by FLIPR analysis
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Copy BDB DOI
Target
Transient receptor potential cation channel subfamily A member 1
(Homo sapiens (Human))
Ferrara University
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.35E+8nM
Assay Description:
Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assay
More data for this Ligand-Target Pair
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In Depth
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Copy BDB DOI
Target
Transient receptor potential cation channel subfamily A member 1
(Homo sapiens (Human))
Ferrara University
Curated by
ChEMBL
Ligand
BDBM26739
(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 2.45E+4nM
Assay Description:
Agonist activity at GDH-tagged human TRPA1 receptor expressed in HEK293F cells assessed as increase in intracellular Ca2+ concentration by FLIPR assa...
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