Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50216321((1R,4R)-2-(5-aminocarbonyl-3-pyridinyl)-2,5-diazab...)
Affinity DataEC50:  2.80E+4nMAssay Description:Agonist activity at alpha-4-beta-2 in IMR-32cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50216321((1R,4R)-2-(5-aminocarbonyl-3-pyridinyl)-2,5-diazab...)
Affinity DataEC50:  2.80E+4nMAssay Description:Agonist activity at alpha-4-beta-2 in IMR-32cells assessed as calcium influx by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed