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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by
ChEMBL
Ligand
BDBM50208758
((RS)-2-amino-[1-hydroxy-5-(3-phenylpropyl)-4-pyraz...)
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Affinity Data
Ki: 6.70E+4nM
Assay Description:
Antagonist activity at rat mGluR2 receptor expressed in CHO cells assessed as effect on intracellular cAMP level
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
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Target
Metabotropic glutamate receptor 1
(RAT)
The Danish University Of Pharmaceutical Sciences
Curated by
ChEMBL
Ligand
BDBM50208758
((RS)-2-amino-[1-hydroxy-5-(3-phenylpropyl)-4-pyraz...)
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Affinity Data
Ki: 2.60E+5nM
Assay Description:
Antagonist activity at rat mGluR1a receptor expressed in CHO cells assessed as effect on intracellular calcium level
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
The Danish University Of Pharmaceutical Sciences
Curated by
ChEMBL
Ligand
BDBM50208758
((RS)-2-amino-[1-hydroxy-5-(3-phenylpropyl)-4-pyraz...)
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Agonist activity at rat mGluR4 receptor expressed in CHO cells assessed as effect on intracellular cAMP level
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI