Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Endoplasmic reticulum aminopeptidase 2
(Homo sapiens (Human))
Wroclaw University Of Technology
Curated by
ChEMBL
Ligand
BDBM50170896
(CHEMBL3805251)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.03E+4nM
Assay Description:
Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Aminopeptidase N
(Homo sapiens (Human))
Wroclaw University Of Technology
Curated by
ChEMBL
Ligand
BDBM50170896
(CHEMBL3805251)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.35E+4nM
Assay Description:
Inhibition of recombinant human alanyl aminopeptidase M1 using Ala-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition mea...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Aminopeptidase N
(Sus scrofa (Pig))
Wroclaw University Of Technology
Curated by
ChEMBL
Ligand
BDBM50170896
(CHEMBL3805251)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.77E+4nM
Assay Description:
Inhibition of pig kidney alanyl aminopeptidase M1 using Ala-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition measured f...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Cytosol aminopeptidase [33-68,L62W]
(Sus scrofa (Pig))
Wroclaw University Of Technology
Curated by
ChEMBL
Ligand
BDBM50170896
(CHEMBL3805251)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.40E+5nM
Assay Description:
Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Endoplasmic reticulum aminopeptidase 1
(Homo sapiens (Human))
Wroclaw University Of Technology
Curated by
ChEMBL
Ligand
BDBM50170896
(CHEMBL3805251)
Copy SMILES
Copy InChI
Affinity Data
Ki: >2.50E+5nM
Assay Description:
Inhibition of recombinant human ERAP1 using L-AMC as substrate measured for 15 to 30 mins by fluorescence analysis
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI