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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
15
hits in this display
Target
Glutamate receptor 4
(Rattus norvegicus)
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
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Affinity Data
Ki: 0.200nM
Assay Description:
Displacement of [3H]AMPA from rat recombinant GluR4 expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Glutamate receptor 3
(RAT)
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
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Affinity Data
Ki: 0.390nM
Assay Description:
Displacement of [3H]AMPA from rat recombinant GluR3 expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Glutamate receptor 2
(Rattus norvegicus)
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
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Affinity Data
Ki: 0.75nM
Assay Description:
Displacement of [3H]AMPA from rat recombinant GluR2 expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Glutamate receptor 1
(Rattus norvegicus (Rat))
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
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Affinity Data
Ki: 7.70nM
Assay Description:
Displacement of [3H]AMPA from rat recombinant GluR1 expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor ionotropic, kainate 2
(Rattus norvegicus)
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
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Affinity Data
Ki: 39nM
Assay Description:
Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor ionotropic, kainate 1
(RAT)
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
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Affinity Data
Ki: 58nM
Assay Description:
Displacement of [3H]SYM 2081 from rat recombinant GluR5 expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor 4
(Rattus norvegicus)
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
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Copy InChI
Affinity Data
Ki: 200nM
Assay Description:
Displacement of (RS)-[3H]AMPA from recombinant rat GluA4 expressed in baculovirus infected Sf9 insect cell membranes
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor 3
(RAT)
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 390nM
Assay Description:
Displacement of (RS)-[3H]AMPA from recombinant rat GluA3 expressed in baculovirus infected Sf9 insect cell membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor 2
(Rattus norvegicus)
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 750nM
Assay Description:
Displacement of (RS)-[3H]AMPA from recombinant rat GluA2(R) expressed in baculovirus infected Sf9 insect cell membranes
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor 1
(Rattus norvegicus (Rat))
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 7.70E+3nM
Assay Description:
Displacement of (RS)-[3H]AMPA from recombinant rat GluA1 expressed in baculovirus infected Sf9 insect cell membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor 3
(Homo sapiens (Human))
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
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Affinity Data
EC50: 1.00E+6nM
Assay Description:
Agonist activity at GluR3 expressed in HEK293 cells by Fluo-4/Ca2+ assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor 4
(Homo sapiens (Human))
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
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Copy InChI
Affinity Data
EC50: 4.90E+5nM
Assay Description:
Agonist activity at GluR4 expressed in Xenopus oocyte cells S-Glutamate
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor 1
(Homo sapiens (Human))
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 3.00E+6nM
Assay Description:
Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor 4
(Homo sapiens (Human))
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 7.50E+4nM
Assay Description:
Agonist activity at GluR4 expressed in HEK293 cells by Fluo-4/Ca2+ assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glutamate receptor 2
(Homo sapiens (Human))
University Of Copenhagen
Curated by
ChEMBL
Ligand
BDBM50211399
((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >3.00E+6nM
Assay Description:
Agonist activity at GluR2Q expressed in HEK293 cells by Fluo-4/Ca2+ assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI