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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
MAP kinase-activated protein kinase 2 [41-364]
(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Ligand
BDBM30284
(indole-based 6-membered lactam, (R)-4a)
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Affinity Data
IC50: 320nM
pH: 7.6 T: 2°C
Assay Description:
Diluted compounds and activated GST-MK2 were incubated in neutravidin coated plates (Pierce) in reaction buffer containing biotinylated GST-LSP1 and ...
More data for this Ligand-Target Pair
Target Info
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MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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Article
PubMed
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Target
Ribosomal protein S6 kinase alpha-3
(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM30284
(indole-based 6-membered lactam, (R)-4a)
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Affinity Data
IC50: 970nM
Assay Description:
Inhibition of RSK2 phosphorylation by luminescence assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI