Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 35 hits in this display
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
Ki: 1.60nMAssay Description:Binding affinity was determined by measuring the ability to displace [125I]SCH-23982 from Dopamine receptor D1 in rat caudate (in vitro)More data for this Ligand-Target Pair
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
Ki: 1.60nMAssay Description:Binding affinity was determined by measuring the ability to displace [125I]SCH-23982 from Dopamine receptor D1 in rat caudate (in vitro)More data for this Ligand-Target Pair
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
Ki: 776nMAssay Description:Binding affinity was determined by measuring the ability to displace [125I]N-(p-aminophenethyl)-spiroperidol from Dopamine receptor D2 in rat caudate...More data for this Ligand-Target Pair
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
Ki: 776nMAssay Description:Binding affinity was determined by measuring the ability to displace [125I]N-(p-aminophenethyl)-spiroperidol from Dopamine receptor D2 in rat caudate...More data for this Ligand-Target Pair
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
Ki: 807nMAssay Description:Binding affinity was determined by measuring the ability to displace [125I]N-(p-aminophenethyl)-spiroperidol from Dopamine receptor D2 in rat caudate...More data for this Ligand-Target Pair
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
Ki: 2.55E+3nMAssay Description:Binding affinity of the compound towards 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand in competitive binding assayMore data for this Ligand-Target Pair
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
Ki: 4.94E+3nMAssay Description:Concentration required to inhibit 50% dopamine receptor D2 in a cell free homogenate of intermediate lobe of pituitary glandMore data for this Ligand-Target Pair
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
Ki: 9.30E+3nMAssay Description:Binding affinity of the compound towards 5-hydroxytryptamine 1C receptor using [125 I]-SCH23982 as radioligand in competitive binding assayMore data for this Ligand-Target Pair
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
Ki: >1.00E+4nMAssay Description:Binding affinity of the compound towards beta-1 adrenergic receptor using [3H]-iodocyanopindolol as radioligand in competitive binding assayMore data for this Ligand-Target Pair
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
Ki: >1.00E+4nMAssay Description:Binding affinity of the compound towards beta-1 adrenergic receptor using [3H]-iodocyanopindolol as radioligand in competitive binding assayMore data for this Ligand-Target Pair
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
Ki: >1.00E+4nMAssay Description:Binding affinity of the compound towards 5-hydroxytryptamine 1C receptor using [125 I]-SCH23982 as radioligand in competitive binding assayMore data for this Ligand-Target Pair
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
Ki: 1.08E+4nMAssay Description:Concentration required to inhibit 50% dopamine receptor D2 in a cell free homogenate of intermediate lobe of pituitary glandMore data for this Ligand-Target Pair
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
Ki: 1.81E+4nMAssay Description:Binding affinity of the compound towards 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand in competitive binding assayMore data for this Ligand-Target Pair
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)
EC50: 1.02E+4nMAssay Description:Concentration required to inhibit 50% dopamine receptor D2 in a cell free homogenate of intermediate lobe of pituitary glandMore data for this Ligand-Target Pair
BDBM50007134(1-Aminomethyl-3-phenyl-isochroman-5,6-diol | CHEMB...)
BDBM50007129((1R,3S)-1-Aminomethyl-3-phenyl-isochroman-5,6-diol...)