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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAminopeptidase N(Sus scrofa (Pig))
Shandong University

LigandPNGBDBM235699((2S)-2-[(2S)-3-amino-2-hydroxypropanamido]-3-pheny...)
Affinity DataIC50:  2.49E+5nMAssay Description:The samples and positive controls were serial diluted to various concentrations: 1280 μg/mL, 320 μg/mL, 80 μg/mL, and 20 μg/mL, 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Shandong University

LigandPNGBDBM235699((2S)-2-[(2S)-3-amino-2-hydroxypropanamido]-3-pheny...)
Affinity DataIC50:  7.10E+5nMpH: 8.5 T: 2°CAssay Description:The compound samples were assayed for inhibitory activity against MMP-2 in 96-well microplates using succinylated gelatin as the substrate. The compo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed