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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
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Target
Amiloride-sensitive amine oxidase [copper-containing]
(Homo sapiens (Human))
Boehringer Ingelheim International
US Patent
Ligand
BDBM220885
(US9302986, 9)
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Affinity Data
IC50: <1.00E+3nM
pH: 7.4 T: 2°C
Assay Description:
Recombinant human DAO (2.4 μg/mL) was used as source of DAO enzyme activities. The assay was performed as described in the method for human SSAO/V...
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Target Info
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antibodypedia
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US Patent
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Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
Boehringer Ingelheim International
US Patent
Ligand
BDBM220885
(US9302986, 9)
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Affinity Data
IC50: >1.00E+4nM
pH: 7.4 T: 2°C
Assay Description:
Recombinant human MAO-B (0.06 mg/mL; Sigma Aldrich) was used as source of MAO-B enzyme activities. The assay was performed in a similar way as for hu...
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Target Info
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US Patent
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Target
Membrane primary amine oxidase
(Rattus norvegicus (Rat))
Boehringer Ingelheim International
US Patent
Ligand
BDBM220885
(US9302986, 9)
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Affinity Data
IC50: <1.00E+5nM
pH: 7.4
Assay Description:
Abdominal fat from BALB/c mice, Wistar or Sprague Dawley rats, which are tissues enriched with SSAO/VAP-1-were surgically removed. For every gram of ...
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US Patent
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Target
Membrane primary amine oxidase
(Homo sapiens (Human))
Boehringer Ingelheim International
US Patent
Ligand
BDBM220885
(US9302986, 9)
Copy SMILES
Copy InChI
Affinity Data
IC50: <1.00E+5nM
pH: 7.4
Assay Description:
Briefly, HMEC cell expressing human SSAO/VAP-1 were grown in several 10 cm petri dishes, once the cells reached 100% confluency, cells were harvested...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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PC cid
PC sid
In Depth
Details
US Patent
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