Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50089515(1-Amino-3-phosphono-cyclopent-3-enecarboxylic acid...)
Affinity DataIC50: >1.00E+5nMAssay Description:Agonistic activity of the compound was tested on Human mGlu4a receptor expressed in recombinant mammalian cells by GTPgammaS binding assay; Partial a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50089515(1-Amino-3-phosphono-cyclopent-3-enecarboxylic acid...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration of the compound was tested on Human mGlu4 receptor expressed in recombinant mammalian cells by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50089515(1-Amino-3-phosphono-cyclopent-3-enecarboxylic acid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of forskolin-stimulated cAMP accumulation in CHO cells expressing hmGlu4aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50089515(1-Amino-3-phosphono-cyclopent-3-enecarboxylic acid...)
Affinity DataEC50:  1.70E+4nMAssay Description:Inhibition of forskolin-stimulated cAMP accumulation in CHO cells expressing hmGlu4aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50089515(1-Amino-3-phosphono-cyclopent-3-enecarboxylic acid...)
Affinity DataEC50: >3.00E+5nMAssay Description:Agonistic activity of the compound was tested on Human Metabotropic glutamate receptor 2 expressed in recombinant mammalian cells by GTPgammaS bindin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed