Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50076394(2-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076394(2-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50076394(2-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Affinity DataIC50:  6.30E+5nMAssay Description:Inhibition of the 1S,3R-ACPD stimulation of IP formation by the compound in LLC-PK1 cells expressing Metabotropic glutamate receptor (mGluRla)More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50076394(2-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Affinity DataEC50:  9.30E+3nMAssay Description:Compound was tested for inhibitory binding activity towards metabotropic glutamate receptor (mGluRla) expressed in LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article