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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
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Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM50076394
(2-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
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Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
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Ligand Info
CHEMBL
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In Depth
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Article
PubMed
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Target
Metabotropic glutamate receptor 1
(RAT)
Parc Club Orsay Université
Curated by
ChEMBL
Ligand
BDBM50076394
(2-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
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Affinity Data
IC50: 3.00E+5nM
Assay Description:
Inhibitory activity of the compound against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM50076394
(2-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.30E+5nM
Assay Description:
Inhibition of the 1S,3R-ACPD stimulation of IP formation by the compound in LLC-PK1 cells expressing Metabotropic glutamate receptor (mGluRla)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
Copy BDB DOI
Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
Emory University
Curated by
PDSP K
i
Database
Ligand
BDBM50076394
(2-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 9.30E+3nM
Assay Description:
Compound was tested for inhibitory binding activity towards metabotropic glutamate receptor (mGluRla) expressed in LLC-PK1 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
Copy BDB DOI