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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
MAP kinase-activated protein kinase 2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50162641
(1,3-Diamino-5-hydroxy-9,9a-dihydro-4aH-xanthene-2-...)
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Affinity Data
IC50: 460nM
Assay Description:
Concentration of 50% inhibition by compound towards mitogen activated protein kinase -activated protein kinase 2
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
MAP kinase-activated protein kinase 2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50162641
(1,3-Diamino-5-hydroxy-9,9a-dihydro-4aH-xanthene-2-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7.12E+3nM
Assay Description:
Inhibition of TNFalpha expression in U937 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI